|
---|
α1 | Agonists | |
---|
Antagonists |
-
Abanoquil
-
Ajmalicine
-
Alfuzosin
-
Anisodamine
-
Anisodine
-
Atiprosin
-
Atypical antipsychotics (e.g.,
brexpiprazole,
clozapine,
olanzapine,
quetiapine,
risperidone)
-
Benoxathian
-
Beta blockers (e.g.,
adimolol,
amosulalol,
arotinolol,
carvedilol,
eugenodilol,
labetalol)
-
Buflomedil
-
Bunazosin
-
Corynanthine
-
Dapiprazole
-
Domesticine
-
Doxazosin
-
Ergolines (e.g.,
acetergamine,
ergotamine,
dihydroergotamine,
lisuride,
nicergoline,
terguride)
-
Etoperidone
-
Fenspiride
-
Hydroxyzine
-
Indoramin
-
Ketanserin
-
L-765,314
-
mCPP
-
Mepiprazole
-
Metazosin
-
Monatepil
-
Moxisylyte
-
Naftopidil
-
Nantenine
-
Neldazosin
-
Niaprazine
-
Niguldipine
-
Pardoprunox
-
Pelanserin
-
Perlapine
-
Phendioxan
-
Phenoxybenzamine
-
Phentolamine
-
Phenylpiperazine
antidepressants (e.g.,
hydroxynefazodone,
nefazodone,
trazodone,
triazoledione)
-
Piperoxan
-
Prazosin
-
Quinazosin
-
Quinidine
-
Silodosin
-
Spegatrine
-
Spiperone
-
Talipexole
-
Tamsulosin
-
Terazosin
-
Tiodazosin
-
Tolazoline
-
Tetracyclic antidepressants (e.g.,
amoxapine,
maprotiline,
mianserin)
-
Tricyclic antidepressants (e.g.,
amitriptyline,
clomipramine,
doxepin,
imipramine,
trimipramine)
-
Trimazosin
-
Typical antipsychotics (e.g.,
chlorpromazine,
fluphenazine,
loxapine,
thioridazine)
-
Urapidil
-
WB-4101
-
Zolertine
|
---|
|
---|
α2 | Agonists | |
---|
Antagonists |
-
1-PP
-
Adimolol
-
Amesergide
-
Aptazapine
-
Atipamezole
-
Atypical antipsychotics (e.g.,
asenapine,
brexpiprazole,
clozapine,
lurasidone,
olanzapine,
paliperidone,
quetiapine,
risperidone,
zotepine)
-
Azapirones (e.g.,
buspirone,
gepirone,
ipsapirone,
tandospirone)
-
BRL-44408
-
Buflomedil
-
Cirazoline
-
Efaroxan
-
Esmirtazapine
-
Fenmetozole
-
Fluparoxan
-
Idazoxan
-
Ketanserin
-
Lisuride
-
mCPP
-
Mianserin
-
Mirtazapine
-
NAN-190
-
Pardoprunox
-
Phentolamine
-
Phenoxybenzamine
-
Piperoxan
-
Piribedil
-
Rauwolscine
-
Rotigotine
-
Setiptiline
-
Spegatrine
-
Spiroxatrine
-
Sunepitron
-
Terguride
-
Tolazoline
-
Typical antipsychotics (e.g.,
chlorpromazine,
fluphenazine,
loxapine,
thioridazine)
-
Yohimbine
|
---|
|
---|
β | |
---|
|
|
---|
MT1Tooltip Melatonin receptor 1 | |
---|
MT2Tooltip Melatonin receptor 2 | |
---|
Unsorted | |
---|
|
|
---|
5-HT1 |
5-HT1A |
- Agonists:
8-OH-DPAT
-
Adatanserin
-
Amphetamine
-
Antidepressants (e.g.,
etoperidone,
hydroxynefazodone,
nefazodone,
trazodone,
triazoledione,
vilazodone,
vortioxetine)
-
Atypical antipsychotics (e.g.,
aripiprazole,
asenapine,
brexpiprazole,
cariprazine,
clozapine,
lurasidone,
quetiapine,
ziprasidone)
-
Azapirones (e.g.,
buspirone,
eptapirone,
gepirone,
perospirone,
tandospirone)
-
Bay R 1531
-
Befiradol
-
BMY-14802
-
Cannabidiol
-
Dimemebfe
-
Dopamine
-
Ebalzotan
-
Eltoprazine
-
Enciprazine
-
Ergolines (e.g.,
bromocriptine,
cabergoline,
dihydroergotamine,
ergotamine,
lisuride,
LSD,
methylergometrine (methylergonovine),
methysergide,
pergolide)
-
F-11,461
-
F-12826
-
F-13714
-
F-14679
-
F-15063
-
F-15,599
-
Flesinoxan
-
Flibanserin
-
Flumexadol
-
Hypidone
-
Lesopitron
-
LY-293284
-
LY-301317
-
mCPP
-
MKC-242
-
Naluzotan
-
NBUMP
-
Osemozotan
-
Oxaflozane
-
Pardoprunox
-
Piclozotan
-
Rauwolscine
-
Repinotan
-
Roxindole
-
RU-24,969
-
S-14,506
-
S-14671
-
S-15535
-
Sarizotan
-
Serotonin (5-HT)
-
SSR-181507
-
Sunepitron
-
Tryptamines (e.g.,
5-CT,
5-MeO-DMT,
5-MT,
bufotenin,
DMT,
indorenate,
N-Me-5-HT,
psilocin,
psilocybin)
-
TGBA01AD
-
U-92,016-A
-
Urapidil
-
Vilazodone
-
Xaliproden
-
Yohimbine
|
- Antagonists:
Atypical antipsychotics (e.g.,
iloperidone,
risperidone,
sertindole)
-
AV965
-
Beta blockers (e.g.,
alprenolol,
carteolol,
cyanopindolol,
iodocyanopindolol,
isamoltane,
oxprenolol,
penbutolol,
pindobind,
pindolol,
propranolol,
tertatolol)
-
BMY-7,378
-
CSP-2503
-
Dotarizine
-
Ergolines (e.g.,
metergoline)
-
FCE-24379
-
Flopropione
-
GR-46611
-
Isamoltane
-
Lecozotan
-
Mefway
-
Metitepine (methiothepin)
-
MIN-117 (WF-516)
-
MPPF
-
NAN-190
-
Robalzotan
-
S-15535
-
SB-649,915
-
SDZ 216-525
-
Spiperone
-
Spiramide
-
Spiroxatrine
-
UH-301
-
WAY-100135
-
WAY-100635
-
Xylamidine
| |
|
---|
5-HT1B |
- Agonists:
Anpirtoline
-
CGS-12066A
-
CP-93129
-
CP-94253
-
CP-122,288
-
CP-135807
-
Eltoprazine
-
Ergolines (e.g.,
bromocriptine,
dihydroergotamine,
ergotamine,
methylergometrine (methylergonovine),
methysergide,
pergolide)
-
mCPP
-
RU-24,969
-
Serotonin (5-HT)
-
Triptans (e.g.,
avitriptan,
donitriptan,
eletriptan,
sumatriptan,
zolmitriptan)
-
TFMPP
-
Tryptamines (e.g.,
5-BT,
5-CT,
5-MT,
DMT)
-
Vortioxetine
| | |
|
---|
5-HT1D |
- Agonists:
CP-122,288
-
CP-135807
-
CP-286601
-
Ergolines (e.g.,
bromocriptine,
cabergoline,
dihydroergotamine,
ergotamine,
LSD,
methysergide)
-
GR-46611
-
L-694247
-
L-772405
-
mCPP
-
PNU-109291
-
PNU-142633
-
Serotonin (5-HT)
-
TGBA01AD
-
Triptans (e.g.,
almotriptan,
avitriptan,
donitriptan,
eletriptan,
frovatriptan,
naratriptan,
rizatriptan,
sumatriptan,
zolmitriptan)
-
Tryptamines (e.g.,
5-BT,
5-CT,
5-Et-DMT,
5-MT,
5-(nonyloxy)tryptamine,
DMT)
| | |
|
---|
5-HT1E | |
---|
5-HT1F | |
---|
|
---|
5-HT2 |
5-HT2A |
- Agonists: 25H/NB series (e.g.,
25I-NBF,
25I-NBMD,
25I-NBOH,
25I-NBOMe,
25B-NBOMe,
25C-NBOMe,
25TFM-NBOMe,
2CBCB-NBOMe,
25CN-NBOH,
2CBFly-NBOMe)
-
2Cs (e.g.,
2C-B,
2C-E,
2C-I,
2C-T-2,
2C-T-7,
2C-T-21)
-
2C-B-FLY
-
2CB-Ind
-
5-Methoxytryptamines (
5-MeO-DET,
5-MeO-DiPT,
5-MeO-DMT,
5-MeO-DPT,
5-MT)
-
α-Alkyltryptamines (e.g.,
5-Cl-αMT,
5-Fl-αMT,
5-MeO-αET,
5-MeO-αMT,
α-Me-5-HT,
αET,
αMT)
-
AL-34662
-
AL-37350A
-
Bromo-DragonFLY
-
Dimemebfe
-
DMBMPP
-
DOx (e.g.,
DOB,
DOC,
DOI,
DOM)
-
Efavirenz
-
Ergolines (e.g.,
1P-LSD,
ALD-52,
bromocriptine,
cabergoline,
ergine (LSA),
ergometrine (ergonovine),
ergotamine,
lisuride,
LA-SS-Az,
LSB,
LSD,
LSD-Pip,
LSH,
LSP,
methylergometrine (methylergonovine),
pergolide)
-
Flumexadol
-
IHCH-7113
-
Jimscaline
-
Lorcaserin
-
MDxx (e.g.,
MDA (tenamfetamine),
MDMA (midomafetamine),
MDOH,
MMDA)
-
O-4310
-
Oxaflozane
-
PHA-57378
-
PNU-22394
-
PNU-181731
-
RH-34
-
SCHEMBL5334361
-
Phenethylamines (e.g.,
lophophine,
mescaline)
-
Piperazines (e.g.,
BZP,
quipazine,
TFMPP)
-
Serotonin (5-HT)
-
TCB-2
-
TFMFly
-
Tryptamines (e.g.,
5-BT,
5-CT,
bufotenin,
DET,
DiPT,
DMT,
DPT,
psilocin,
psilocybin,
tryptamine)
|
- Antagonists:
5-I-R91150
-
5-MeO-NBpBrT
-
AC-90179
-
Adatanserin
-
Altanserin
-
Antihistamines (e.g.,
cyproheptadine,
hydroxyzine,
ketotifen,
perlapine)
-
AMDA
-
Atypical antipsychotics (e.g.,
amperozide,
aripiprazole,
asenapine,
blonanserin,
brexpiprazole,
carpipramine,
clocapramine,
clorotepine,
clozapine,
fluperlapine,
gevotroline,
iloperidone,
lurasidone,
melperone,
mosapramine,
ocaperidone,
olanzapine,
paliperidone,
quetiapine,
risperidone,
sertindole,
zicronapine,
ziprasidone,
zotepine)
-
Chlorprothixene
-
Cinanserin
-
CSP-2503
-
Deramciclane
-
Dotarizine
-
Eplivanserin
-
Ergolines (e.g.,
amesergide,
LY-53857,
LY-215,840,
mesulergine,
metergoline,
methysergide,
sergolexole)
-
Fananserin
-
Flibanserin
-
Glemanserin
-
Irindalone
-
Ketanserin
-
KML-010
-
Landipirdine
-
LY-393558
-
mCPP
-
Medifoxamine
-
Metitepine (methiothepin)
-
MIN-117 (WF-516)
-
Naftidrofuryl
-
Nantenine
-
Nelotanserin
-
Opiranserin (VVZ-149)
-
Pelanserin
-
Phenoxybenzamine
-
Pimavanserin
-
Pirenperone
-
Pizotifen
-
Pruvanserin
-
Rauwolscine
-
Ritanserin
-
Roluperidone
-
S-14671
-
Sarpogrelate
-
Serotonin antagonists and reuptake inhibitors (e.g.,
etoperidone,
hydroxynefazodone,
lubazodone,
mepiprazole,
nefazodone,
triazoledione,
trazodone)
-
SR-46349B
-
TGBA01AD
-
Teniloxazine
-
Temanogrel
-
Tetracyclic antidepressants (e.g.,
amoxapine,
aptazapine,
esmirtazapine,
maprotiline,
mianserin,
mirtazapine)
-
Tricyclic antidepressants (e.g.,
amitriptyline)
-
Typical antipsychotics (e.g.,
chlorpromazine,
fluphenazine,
haloperidol,
loxapine,
perphenazine,
pimozide,
pipamperone,
prochlorperazine,
setoperone,
spiperone,
spiramide,
thioridazine,
thiothixene,
trifluoperazine)
-
Volinanserin
-
Xylamidine
-
Yohimbine
| |
|
---|
5-HT2B |
- Agonists:
4-Methylaminorex
-
Aminorex
-
Amphetamines (e.g.,
chlorphentermine,
cloforex,
dexfenfluramine,
fenfluramine,
levofenfluramine,
norfenfluramine)
-
BW-723C86
-
DOx (e.g.,
DOB,
DOC,
DOI,
DOM)
-
Ergolines (e.g.,
cabergoline,
dihydroergocryptine,
dihydroergotamine,
ergotamine,
methylergometrine (methylergonovine),
methysergide,
pergolide)
-
Lorcaserin
-
MDxx (e.g.,
MDA (tenamfetamine),
MDMA (midomafetamine),
MDOH,
MMDA)
-
Piperazines (e.g.,
TFMPP)
-
PNU-22394
-
Ro60-0175
-
Serotonin (5-HT)
-
Tryptamines (e.g.,
5-BT,
5-CT,
5-MT,
α-Me-5-HT,
bufotenin,
DET,
DiPT,
DMT,
DPT,
psilocin,
psilocybin,
tryptamine)
|
- Antagonists:
Agomelatine
-
Atypical antipsychotics (e.g.,
amisulpride,
aripiprazole,
asenapine,
brexpiprazole,
cariprazine,
clozapine,
N-desalkylquetiapine (norquetiapine),
N-desmethylclozapine (norclozapine),
olanzapine,
pipamperone,
quetiapine,
risperidone,
ziprasidone)
-
Cyproheptadine
-
EGIS-7625
-
Ergolines (e.g.,
amesergide,
bromocriptine,
lisuride,
LY-53857,
LY-272015,
mesulergine)
-
Ketanserin
-
LY-393558
-
mCPP
-
Metadoxine
-
Metitepine (methiothepin)
-
Pirenperone
-
Pizotifen
-
Propranolol
-
PRX-08066
-
Rauwolscine
-
Ritanserin
-
RS-127445
-
Sarpogrelate
-
SB-200646
-
SB-204741
-
SB-206553
-
SB-215505
-
SB-221284
-
SB-228357
-
SDZ SER-082
-
Tegaserod
-
Tetracyclic antidepressants (e.g.,
amoxapine,
mianserin,
mirtazapine)
-
Trazodone
-
Typical antipsychotics (e.g.,
chlorpromazine)
-
TIK-301
-
Yohimbine
| |
|
---|
5-HT2C |
- Agonists:
2Cs (e.g.,
2C-B,
2C-E,
2C-I,
2C-T-2,
2C-T-7,
2C-T-21)
-
5-Methoxytryptamines (
5-MeO-DET,
5-MeO-DiPT,
5-MeO-DMT,
5-MeO-DPT,
5-MT)
-
α-Alkyltryptamines (e.g.,
5-Cl-αMT,
5-Fl-αMT,
5-MeO-αET,
5-MeO-αMT,
α-Me-5-HT,
αET,
αMT)
-
A-372159
-
AL-38022A
-
Alstonine
-
CP-809101
-
Dimemebfe
-
DOx (e.g.,
DOB,
DOC,
DOI,
DOM)
-
Ergolines (e.g.,
ALD-52,
cabergoline,
dihydroergotamine,
ergine (LSA),
ergotamine,
lisuride,
LA-SS-Az,
LSB,
LSD,
LSD-Pip,
LSH,
LSP,
pergolide)
-
Flumexadol
-
Lorcaserin
-
MDxx (e.g.,
MDA (tenamfetamine),
MDMA (midomafetamine),
MDOH,
MMDA)
-
MK-212
-
ORG-12962
-
ORG-37684
-
Oxaflozane
-
PHA-57378
-
Phenethylamines (e.g.,
lophophine,
mescaline)
-
Piperazines (e.g.,
aripiprazole,
BZP,
mCPP,
quipazine,
TFMPP)
-
PNU-22394
-
PNU-181731
-
Ro60-0175
-
Ro60-0213
-
Serotonin (5-HT)
-
Tryptamines (e.g.,
5-BT,
5-CT,
bufotenin,
DET,
DiPT,
DMT,
DPT,
psilocin,
psilocybin,
tryptamine)
-
Vabicaserin
-
WAY-629
-
WAY-161503
-
YM-348
|
- Antagonists:
Adatanserin
-
Agomelatine
-
Atypical antipsychotics (e.g.,
asenapine,
clorotepine,
clozapine,
fluperlapine,
iloperidone,
melperone,
olanzapine,
paliperidone,
quetiapine,
risperidone,
sertindole,
ziprasidone,
zotepine)
-
Captodiame
-
CEPC
-
Cinanserin
-
Cyproheptadine
-
Deramciclane
-
Desmetramadol
-
Dotarizine
-
Eltoprazine
-
Ergolines (e.g.,
amesergide,
bromocriptine,
LY-53857,
LY-215,840,
mesulergine,
metergoline,
methysergide,
sergolexole)
-
Etoperidone
-
Fluoxetine
-
FR-260010
-
Irindalone
-
Ketanserin
-
Ketotifen
-
Latrepirdine (dimebolin)
-
Medifoxamine
-
Metitepine (methiothepin)
-
Nefazodone
-
Pirenperone
-
Pizotifen
-
Propranolol
-
Ritanserin
-
RS-102221
-
S-14671
-
SB-200646
-
SB-206553
-
SB-221284
-
SB-228357
-
SB-242084
-
SB-243213
-
SDZ SER-082
-
Tedatioxetine
-
Tetracyclic antidepressants (e.g.,
amoxapine,
aptazapine,
esmirtazapine,
maprotiline,
mianserin,
mirtazapine)
-
TIK-301
-
Tramadol
-
Trazodone
-
Tricyclic antidepressants (e.g.,
amitriptyline,
nortriptyline)
-
Typical antipsychotics (e.g.,
chlorpromazine,
loxapine,
pimozide,
pipamperone,
thioridazine)
-
Xylamidine
| |
|
---|
|
---|
5-HT3–
7 |
5-HT3 |
- Agonists:
Alcohols (e.g.,
butanol,
ethanol (alcohol),
trichloroethanol)
-
m-CPBG
-
Phenylbiguanide
-
Piperazines (e.g.,
BZP,
mCPP,
quipazine)
-
RS-56812
-
Serotonin (5-HT)
-
SR-57227
-
SR-57227A
-
Tryptamines (e.g.,
2-Me-5-HT,
5-CT,
bufotenidine (5-HTQ))
-
Volatiles/gases (e.g.,
halothane,
isoflurane,
toluene,
trichloroethane)
-
YM-31636
|
- Antagonists:
Alosetron
-
Anpirtoline
-
Arazasetron
-
AS-8112
-
Atypical antipsychotics (e.g.,
clozapine,
olanzapine,
quetiapine)
-
Azasetron
-
Batanopride
-
Bemesetron (MDL-72222)
-
Bupropion
-
Cilansetron
-
CSP-2503
-
Dazopride
-
Dolasetron
-
Galanolactone
-
Granisetron
-
Hydroxybupropion
-
Lerisetron
-
Memantine
-
Ondansetron
-
Palonosetron
-
Ramosetron
-
Renzapride
-
Ricasetron
-
Tedatioxetine
-
Tetracyclic antidepressants (e.g.,
amoxapine,
mianserin,
mirtazapine)
-
Thujone
-
Tropanserin
-
Tropisetron
-
Typical antipsychotics (e.g.,
loxapine)
-
Volatiles/gases (e.g.,
nitrous oxide,
sevoflurane,
xenon)
-
Vortioxetine
-
Zacopride
-
Zatosetron
| |
|
---|
5-HT4 | |
---|
5-HT5A | |
---|
5-HT6 |
- Agonists:
Ergolines (e.g.,
dihydroergocryptine,
dihydroergotamine,
ergotamine,
lisuride,
LSD,
mesulergine,
metergoline,
methysergide)
-
Hypidone
-
Serotonin (5-HT)
-
Tryptamines (e.g.,
2-Me-5-HT,
5-BT,
5-CT,
5-MT,
Bufotenin,
E-6801,
E-6837,
EMD-386088,
EMDT,
LY-586713,
N-Me-5-HT,
ST-1936,
tryptamine)
-
WAY-181187
-
WAY-208466
|
- Antagonists:
ABT-354
-
Atypical antipsychotics (e.g.,
aripiprazole,
asenapine,
clorotepine,
clozapine,
fluperlapine,
iloperidone,
olanzapine,
tiospirone)
-
AVN-101
-
AVN-211
-
AVN-322
-
AVN-397
-
BGC20-760
-
BVT-5182
-
BVT-74316
-
Cerlapirdine
-
EGIS-12,233
-
GW-742457
-
Idalopirdine
-
Ketanserin
-
Landipirdine
-
Latrepirdine (dimebolin)
-
Masupirdine
-
Metitepine (methiothepin)
-
MS-245
-
PRX-07034
-
Ritanserin
-
Ro 04-6790
-
Ro 63-0563
-
SB-258585
-
SB-271046
-
SB-357134
-
SB-399885
-
SB-742457
-
Tetracyclic antidepressants (e.g.,
amoxapine,
mianserin)
-
Tricyclic antidepressants (e.g.,
amitriptyline,
clomipramine,
doxepin,
nortriptyline)
-
Typical antipsychotics (e.g.,
chlorpromazine,
loxapine)
| |
|
---|
5-HT7 | |
- Antagonists:
Atypical antipsychotics (e.g.,
amisulpride,
aripiprazole,
asenapine,
brexpiprazole,
clorotepine,
clozapine,
fluperlapine,
olanzapine,
risperidone,
sertindole,
tiospirone,
ziprasidone,
zotepine)
-
Butaclamol
-
DR-4485
-
EGIS-12,233
-
Ergolines (e.g.,
2-Br-LSD (BOL-148),
amesergide,
bromocriptine,
cabergoline,
dihydroergotamine,
ergotamine,
LY-53857,
LY-215,840,
mesulergine,
metergoline,
methysergide,
sergolexole)
-
JNJ-18038683
-
Ketanserin
-
LY-215,840
-
Metitepine (methiothepin)
-
Ritanserin
-
SB-258719
-
SB-258741
-
SB-269970
-
SB-656104
-
SB-656104A
-
SB-691673
-
SLV-313
-
SLV-314
-
Spiperone
-
SSR-181507
-
Tetracyclic antidepressants (e.g.,
amoxapine,
maprotiline,
mianserin,
mirtazapine)
-
Tricyclic antidepressants (e.g.,
amitriptyline,
clomipramine,
imipramine)
-
Typical antipsychotics (e.g.,
acetophenazine,
chlorpromazine,
chlorprothixene,
fluphenazine,
loxapine,
pimozide)
-
Vortioxetine
| |
|
---|
|
---|
|
|