Clinical data | |
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Routes of administration | Oral |
ATC code |
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Identifiers | |
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CAS Number | |
PubChem CID | |
IUPHAR/BPS | |
ChemSpider | |
UNII | |
ChEMBL | |
Chemical and physical data | |
Formula | C20H29NO2 |
Molar mass | 315.457 g·mol−1 |
3D model ( JSmol) | |
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Bremazocine is a κ-opioid receptor agonist related to pentazocine. It has potent and long-lasting analgesic and diuretic effects. [1] It has 200 times the activity of morphine, but appears to have no addictive properties and does not depress breathing. [2] The crystal structure of bremazocine was determined in 1984 [3]
Psychedelics ( 5-HT2A agonists) |
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Dissociatives ( NMDAR antagonists) |
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Deliriants ( mAChR antagonists) |
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Others |
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μ-opioid (MOR) |
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δ-opioid (DOR) |
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κ-opioid (KOR) |
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Nociceptin (NOP) |
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Others |
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Clinical data | |
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Routes of administration | Oral |
ATC code |
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Identifiers | |
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CAS Number | |
PubChem CID | |
IUPHAR/BPS | |
ChemSpider | |
UNII | |
ChEMBL | |
Chemical and physical data | |
Formula | C20H29NO2 |
Molar mass | 315.457 g·mol−1 |
3D model ( JSmol) | |
|
Bremazocine is a κ-opioid receptor agonist related to pentazocine. It has potent and long-lasting analgesic and diuretic effects. [1] It has 200 times the activity of morphine, but appears to have no addictive properties and does not depress breathing. [2] The crystal structure of bremazocine was determined in 1984 [3]
Opioids |
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NSAIDs |
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Ion channel modulators |
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Others | |||||||||||||||||
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Psychedelics ( 5-HT2A agonists) |
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Dissociatives ( NMDAR antagonists) |
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Deliriants ( mAChR antagonists) |
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Others |
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μ-opioid (MOR) |
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δ-opioid (DOR) |
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κ-opioid (KOR) |
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Nociceptin (NOP) |
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Others |
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