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ChEMBL | |
Chemical and physical data | |
Formula | C26H38O2 |
Molar mass | 382.588 g·mol−1 |
3D model ( JSmol) | |
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AM-855 (part of the AM cannabinoid series) is an analgesic drug which is a cannabinoid agonist. It is a derivative of Δ8 Tetrahydrocannabinol with a conformationally restricted side chain which has been bound into a fourth ring fused to the aromatic A-ring of the cannabinoid skeleton. AM-855 is an agonist at both CB1 and CB2 with moderate selectivity for CB1, with a Ki of 22.3 nM at CB1 and 58.6 nM at CB2. [1]
This cannabinoid related article is a stub. You can help Wikipedia by expanding it. |
Identifiers | |
---|---|
| |
CAS Number | |
PubChem CID | |
ChemSpider |
|
UNII | |
ChEMBL | |
Chemical and physical data | |
Formula | C26H38O2 |
Molar mass | 382.588 g·mol−1 |
3D model ( JSmol) | |
| |
| |
(verify) |
AM-855 (part of the AM cannabinoid series) is an analgesic drug which is a cannabinoid agonist. It is a derivative of Δ8 Tetrahydrocannabinol with a conformationally restricted side chain which has been bound into a fourth ring fused to the aromatic A-ring of the cannabinoid skeleton. AM-855 is an agonist at both CB1 and CB2 with moderate selectivity for CB1, with a Ki of 22.3 nM at CB1 and 58.6 nM at CB2. [1]
Phytocannabinoids ( comparison) |
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Endocannabinoids |
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Synthetic cannabinoid receptor agonists / neocannabinoids |
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Allosteric CBRTooltip Cannabinoid receptor ligands | |||||||||||||||||||||||||||||||||||||||||||||||||||
Endocannabinoid enhancers (inactivation inhibitors) |
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Anticannabinoids (antagonists/inverse agonists/antibodies) |
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This cannabinoid related article is a stub. You can help Wikipedia by expanding it. |