From Wikipedia, the free encyclopedia
Chemical compound
CP-39,332 is a
drug which acts as a
serotonin-norepinephrine reuptake inhibitor .
[1]
Tametraline (1R ,4S -),
CP-24,442 (1S ,4R -),
CP-22,185 (cis -), and
CP-22,186 (trans -) are
stereoisomers of the compound and show varying effects on
monoamine
reuptake .
[1] None of them were ever marketed.
See also
References
^
a
b
Koe BK (December 1976). "Molecular geometry of inhibitors of the uptake of catecholamines and serotonin in synaptosomal preparations of rat brain". The Journal of Pharmacology and Experimental Therapeutics . 199 (3): 649–61.
PMID
994022 .
SSRIs Tooltip Selective serotonin reuptake inhibitors
SNRIs Tooltip Serotonin–norepinephrine reuptake inhibitors
NRIs Tooltip Norepinephrine reuptake inhibitors
NDRIs Tooltip Norepinephrine–dopamine reuptake inhibitors
NaSSAs Tooltip Noradrenergic and specific serotonergic antidepressants
SARIs Tooltip Serotonin antagonist and reuptake inhibitors
SMS Tooltip Serotonin modulator and stimulators Others
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Non-selective
MAOA Tooltip Monoamine oxidase A -selective
MAOB Tooltip Monoamine oxidase B -selective
DAT Tooltip Dopamine transporter (
DRIs Tooltip Dopamine reuptake inhibitors )
NET Tooltip Norepinephrine transporter (
NRIs Tooltip Norepinephrine reuptake inhibitors )
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SERT Tooltip Serotonin transporter (
SRIs Tooltip Serotonin reuptake inhibitors )
Others:
A-80426
Amoxapine
Antihistamines (e.g.,
brompheniramine ,
chlorphenamine ,
dimenhydrinate ,
diphenhydramine ,
mepyramine (pyrilamine) ,
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Antipsychotics (e.g.,
loxapine ,
ziprasidone )
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ketamine ,
methoxetamine ,
phencyclidine )
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MIN-117 (WF-516)
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