Clinical data | |
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Routes of administration | Oral |
ATC code |
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Legal status | |
Legal status |
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Identifiers | |
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CAS Number | |
PubChem CID | |
ChemSpider | |
UNII | |
ChEMBL | |
CompTox Dashboard ( EPA) | |
ECHA InfoCard | 100.041.153 |
Chemical and physical data | |
Formula | C24H31N3O |
Molar mass | 377.532 g·mol−1 |
3D model ( JSmol) | |
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Famprofazone (Gewodin, Gewolen) is a nonsteroidal anti-inflammatory agent (NSAID) of the pyrazolone series which is available over-the-counter in some countries such as Taiwan. [1] [2] [3] It has analgesic, anti-inflammatory, and antipyretic effects. [1] [2] Famprofazone has been known to produce methamphetamine as an active metabolite, with 15–20% of an oral dose being converted to it. [4] [5] As a result, famprofazone has occasionally been implicated in causing positives on drug tests for amphetamines. [3]
pyrazolones / pyrazolidines | |
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salicylates | |
acetic acid derivatives and related substances | |
oxicams | |
propionic acid derivatives ( profens) |
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n-arylanthranilic acids ( fenamates) | |
COX-2 inhibitors (coxibs) | |
other | |
NSAID combinations | |
Key: underline indicates initially developed first-in-class compound of specific group; #
WHO-Essential Medicines; †
withdrawn drugs; ‡
veterinary use. | |
DRAsTooltip Dopamine releasing agents |
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NRAsTooltip Norepinephrine releasing agents |
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SRAsTooltip Serotonin releasing agents |
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Others |
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CARTooltip Constitutive androstane receptor |
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PXRTooltip Pregnane X receptor |
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Phenethylamines |
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Amphetamines |
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Phentermines |
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Cathinones |
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Phenylisobutylamines | |
Phenylalkylpyrrolidines | |
Catecholamines (and close relatives) |
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Miscellaneous |
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Clinical data | |
---|---|
Routes of administration | Oral |
ATC code |
|
Legal status | |
Legal status |
|
Identifiers | |
| |
CAS Number | |
PubChem CID | |
ChemSpider | |
UNII | |
ChEMBL | |
CompTox Dashboard ( EPA) | |
ECHA InfoCard | 100.041.153 |
Chemical and physical data | |
Formula | C24H31N3O |
Molar mass | 377.532 g·mol−1 |
3D model ( JSmol) | |
|
Famprofazone (Gewodin, Gewolen) is a nonsteroidal anti-inflammatory agent (NSAID) of the pyrazolone series which is available over-the-counter in some countries such as Taiwan. [1] [2] [3] It has analgesic, anti-inflammatory, and antipyretic effects. [1] [2] Famprofazone has been known to produce methamphetamine as an active metabolite, with 15–20% of an oral dose being converted to it. [4] [5] As a result, famprofazone has occasionally been implicated in causing positives on drug tests for amphetamines. [3]
pyrazolones / pyrazolidines | |
---|---|
salicylates | |
acetic acid derivatives and related substances | |
oxicams | |
propionic acid derivatives ( profens) |
|
n-arylanthranilic acids ( fenamates) | |
COX-2 inhibitors (coxibs) | |
other | |
NSAID combinations | |
Key: underline indicates initially developed first-in-class compound of specific group; #
WHO-Essential Medicines; †
withdrawn drugs; ‡
veterinary use. | |
Opioids |
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Ion channel modulators |
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DRAsTooltip Dopamine releasing agents |
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NRAsTooltip Norepinephrine releasing agents |
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SRAsTooltip Serotonin releasing agents |
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Others |
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CARTooltip Constitutive androstane receptor |
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PXRTooltip Pregnane X receptor |
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Phenethylamines |
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Amphetamines |
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Phentermines |
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Cathinones |
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Phenylisobutylamines | |
Phenylalkylpyrrolidines | |
Catecholamines (and close relatives) |
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Miscellaneous |
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