Identifiers | |
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CAS Number |
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PubChem CID | |
ChemSpider | |
UNII |
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Chemical and physical data | |
Formula | C22H28ClNO |
Molar mass | 357.92 g·mol−1 |
3D model ( JSmol) | |
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Setastine (Loderix) is an antihistamine used to treat allergies and rhinitis. [1] [2]
Setastine acts as a highly selective H1 receptor antagonist. [3] It has no anticholinergic, antiadrenergic, or antiserotonergic effects.
Setastine penetrates the blood-brain-barrier poorly so it is only mildly sedating compared to related molecules like diphenhydramine. [3]
Identifiers | |
---|---|
| |
CAS Number |
|
PubChem CID | |
ChemSpider | |
UNII |
|
Chemical and physical data | |
Formula | C22H28ClNO |
Molar mass | 357.92 g·mol−1 |
3D model ( JSmol) | |
|
Setastine (Loderix) is an antihistamine used to treat allergies and rhinitis. [1] [2]
Setastine acts as a highly selective H1 receptor antagonist. [3] It has no anticholinergic, antiadrenergic, or antiserotonergic effects.
Setastine penetrates the blood-brain-barrier poorly so it is only mildly sedating compared to related molecules like diphenhydramine. [3]