Clinical data | |
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ATC code |
|
Pharmacokinetic data | |
Bioavailability | 34% |
Protein binding | 69% |
Elimination half-life | 1.8h |
Identifiers | |
| |
CAS Number | |
ChemSpider | |
ChEMBL | |
Chemical and physical data | |
Formula | C21H23ClN6 |
Molar mass | 394.91 g·mol−1 |
3D model ( JSmol) | |
| |
| |
(what is this?) (verify) |
PF-184563 is a potent, selective non-peptidic antagonist of the V1a receptor. [1] The compound was discovered by Pfizer in its Sandwich, Kent research center, as a potential treatment for dysmenorrhoea, an indication for which V1a antagonists have shown efficacy. [2]
Clinical data | |
---|---|
ATC code |
|
Pharmacokinetic data | |
Bioavailability | 34% |
Protein binding | 69% |
Elimination half-life | 1.8h |
Identifiers | |
| |
CAS Number | |
ChemSpider | |
ChEMBL | |
Chemical and physical data | |
Formula | C21H23ClN6 |
Molar mass | 394.91 g·mol−1 |
3D model ( JSmol) | |
| |
| |
(what is this?) (verify) |
PF-184563 is a potent, selective non-peptidic antagonist of the V1a receptor. [1] The compound was discovered by Pfizer in its Sandwich, Kent research center, as a potential treatment for dysmenorrhoea, an indication for which V1a antagonists have shown efficacy. [2]