From Wikipedia, the free encyclopedia
Medications and dosages used in transgender women [1] [2] [3] [4] [5] [a]
Medication Brand name Type Route Dosage [b]
Estradiol Various Estrogen Oral 2–10 mg/day
Various Estrogen Sublingual 1–8 mg/day
Climara [c] Estrogen TD patch 25–400 μg/day
Divigel [c] Estrogen TD gel 0.5–5 mg/day
Various Estrogen SC implant 50–200 mg every 6–24 mos
Estradiol valerate Progynova Estrogen Oral 2–10 mg/day
Progynova Estrogen Sublingual 1–8 mg/day
Delestrogen [c] Estrogen IM, SC 2–10 mg/ wk or
5–20 mg every 2 wks
Estradiol cypionate Depo-Estradiol Estrogen IM, SC 2–10 mg/wk or
5–20 mg every 2 wks
Estradiol dipropionate Agofollin Estrogen IM, SC 2–10 mg/wk or
5–20 mg every 2 wks
Estradiol benzoate Progynon-B Estrogen IM, SC 0.5–1.5 mg every 2–3 days
Estriol Ovestin [c] Estrogen Oral 4–6 mg/day
Spironolactone Aldactone Antiandrogen Oral 100–400 mg/day
Cyproterone acetate Androcur Antiandrogen;
Progestogen
Oral 5–100 mg/day
Androcur Depot IM 300 mg/month
Bicalutamide Casodex Antiandrogen Oral 25–50 mg/day
Enzalutamide Xtandi Antiandrogen Oral 160 mg/day
GnRH analogue Various GnRH modulator Various Variable
Elagolix Orilissa GnRH antagonist Oral 150 mg/day or
200 mg twice daily
Finasteride Propecia 5αR inhibitor Oral 1–5 mg/day
Dutasteride Avodart 5αR inhibitor Oral 0.25–0.5 mg/day
Progesterone Prometrium [c] Progestogen Oral 100–400 mg/day
Medroxyprogesterone acetate Provera Progestogen Oral 2.5–40 mg/day
Depo-Provera Progestogen IM 150 mg every 3  mos
Depo-SubQ Provera 104 Progestogen SC 104 mg every 3 mos
Hydroxyprogesterone caproate Proluton Progestogen IM 250 mg/wk
Dydrogesterone Duphaston Progestogen Oral 20 mg/day
Drospirenone Slynd Progestogen Oral 3 mg/day
Domperidone [d] Motilium Prolactin releaser Oral 30–80 mg/day [e]
  1. ^ Additional sources: [6] [7] [8] [9] [10] [11] [12] [13] [14] [15] [16] [17] [18] [19] [20] [21] [22] [23] [24] [25] [26] [27] [28] [29] [30] [31] [32] [33] [34] [35] [36]
  2. ^ Lower starting doses may be used in adolescents if being used in combination with a GnRH agonist or antagonist.
  3. ^ a b c d e Also available under other brand names.
  4. ^ For induction of lactation to allow for breastfeeding specifically.
  5. ^ Administered in divided doses.
From Wikipedia, the free encyclopedia
Medications and dosages used in transgender women [1] [2] [3] [4] [5] [a]
Medication Brand name Type Route Dosage [b]
Estradiol Various Estrogen Oral 2–10 mg/day
Various Estrogen Sublingual 1–8 mg/day
Climara [c] Estrogen TD patch 25–400 μg/day
Divigel [c] Estrogen TD gel 0.5–5 mg/day
Various Estrogen SC implant 50–200 mg every 6–24 mos
Estradiol valerate Progynova Estrogen Oral 2–10 mg/day
Progynova Estrogen Sublingual 1–8 mg/day
Delestrogen [c] Estrogen IM, SC 2–10 mg/ wk or
5–20 mg every 2 wks
Estradiol cypionate Depo-Estradiol Estrogen IM, SC 2–10 mg/wk or
5–20 mg every 2 wks
Estradiol dipropionate Agofollin Estrogen IM, SC 2–10 mg/wk or
5–20 mg every 2 wks
Estradiol benzoate Progynon-B Estrogen IM, SC 0.5–1.5 mg every 2–3 days
Estriol Ovestin [c] Estrogen Oral 4–6 mg/day
Spironolactone Aldactone Antiandrogen Oral 100–400 mg/day
Cyproterone acetate Androcur Antiandrogen;
Progestogen
Oral 5–100 mg/day
Androcur Depot IM 300 mg/month
Bicalutamide Casodex Antiandrogen Oral 25–50 mg/day
Enzalutamide Xtandi Antiandrogen Oral 160 mg/day
GnRH analogue Various GnRH modulator Various Variable
Elagolix Orilissa GnRH antagonist Oral 150 mg/day or
200 mg twice daily
Finasteride Propecia 5αR inhibitor Oral 1–5 mg/day
Dutasteride Avodart 5αR inhibitor Oral 0.25–0.5 mg/day
Progesterone Prometrium [c] Progestogen Oral 100–400 mg/day
Medroxyprogesterone acetate Provera Progestogen Oral 2.5–40 mg/day
Depo-Provera Progestogen IM 150 mg every 3  mos
Depo-SubQ Provera 104 Progestogen SC 104 mg every 3 mos
Hydroxyprogesterone caproate Proluton Progestogen IM 250 mg/wk
Dydrogesterone Duphaston Progestogen Oral 20 mg/day
Drospirenone Slynd Progestogen Oral 3 mg/day
Domperidone [d] Motilium Prolactin releaser Oral 30–80 mg/day [e]
  1. ^ Additional sources: [6] [7] [8] [9] [10] [11] [12] [13] [14] [15] [16] [17] [18] [19] [20] [21] [22] [23] [24] [25] [26] [27] [28] [29] [30] [31] [32] [33] [34] [35] [36]
  2. ^ Lower starting doses may be used in adolescents if being used in combination with a GnRH agonist or antagonist.
  3. ^ a b c d e Also available under other brand names.
  4. ^ For induction of lactation to allow for breastfeeding specifically.
  5. ^ Administered in divided doses.

Videos

Youtube | Vimeo | Bing

Websites

Google | Yahoo | Bing

Encyclopedia

Google | Yahoo | Bing

Facebook