Medication | Brand name | Type | Route | Dosage [b] |
---|---|---|---|---|
Estradiol | Various | Estrogen | Oral | 2–10 mg/day |
Various | Estrogen | Sublingual | 1–8 mg/day | |
Climara [c] | Estrogen | TD patch | 25–400 μg/day | |
Divigel [c] | Estrogen | TD gel | 0.5–5 mg/day | |
Various | Estrogen | SC implant | 50–200 mg every 6–24 mos | |
Estradiol valerate | Progynova | Estrogen | Oral | 2–10 mg/day |
Progynova | Estrogen | Sublingual | 1–8 mg/day | |
Delestrogen [c] | Estrogen | IM, SC | 2–10 mg/
wk or 5–20 mg every 2 wks | |
Estradiol cypionate | Depo-Estradiol | Estrogen | IM, SC | 2–10 mg/wk or 5–20 mg every 2 wks |
Estradiol dipropionate | Agofollin | Estrogen | IM, SC | 2–10 mg/wk or 5–20 mg every 2 wks |
Estradiol benzoate | Progynon-B | Estrogen | IM, SC | 0.5–1.5 mg every 2–3 days |
Estriol | Ovestin [c] | Estrogen | Oral | 4–6 mg/day |
Spironolactone | Aldactone | Antiandrogen | Oral | 100–400 mg/day |
Cyproterone acetate | Androcur | Antiandrogen; Progestogen |
Oral | 5–100 mg/day |
Androcur Depot | IM | 300 mg/month | ||
Bicalutamide | Casodex | Antiandrogen | Oral | 25–50 mg/day |
Enzalutamide | Xtandi | Antiandrogen | Oral | 160 mg/day |
GnRH analogue | Various | GnRH modulator | Various | Variable |
Elagolix | Orilissa | GnRH antagonist | Oral | 150 mg/day or 200 mg twice daily |
Finasteride | Propecia | 5αR inhibitor | Oral | 1–5 mg/day |
Dutasteride | Avodart | 5αR inhibitor | Oral | 0.25–0.5 mg/day |
Progesterone | Prometrium [c] | Progestogen | Oral | 100–400 mg/day |
Medroxyprogesterone acetate | Provera | Progestogen | Oral | 2.5–40 mg/day |
Depo-Provera | Progestogen | IM | 150 mg every 3 mos | |
Depo-SubQ Provera 104 | Progestogen | SC | 104 mg every 3 mos | |
Hydroxyprogesterone caproate | Proluton | Progestogen | IM | 250 mg/wk |
Dydrogesterone | Duphaston | Progestogen | Oral | 20 mg/day |
Drospirenone | Slynd | Progestogen | Oral | 3 mg/day |
Domperidone [d] | Motilium | Prolactin releaser | Oral | 30–80 mg/day [e] |
|
When we prescribed estradiol, we preferred sublingual estradiol valerate instead of the oral form for feminizing HT since prior researchers have reported the effectiveness of sublingual administration in maintaining high blood estradiol concentration and low E1/E2 ratio [13].
Medication | Brand name | Type | Route | Dosage [b] |
---|---|---|---|---|
Estradiol | Various | Estrogen | Oral | 2–10 mg/day |
Various | Estrogen | Sublingual | 1–8 mg/day | |
Climara [c] | Estrogen | TD patch | 25–400 μg/day | |
Divigel [c] | Estrogen | TD gel | 0.5–5 mg/day | |
Various | Estrogen | SC implant | 50–200 mg every 6–24 mos | |
Estradiol valerate | Progynova | Estrogen | Oral | 2–10 mg/day |
Progynova | Estrogen | Sublingual | 1–8 mg/day | |
Delestrogen [c] | Estrogen | IM, SC | 2–10 mg/
wk or 5–20 mg every 2 wks | |
Estradiol cypionate | Depo-Estradiol | Estrogen | IM, SC | 2–10 mg/wk or 5–20 mg every 2 wks |
Estradiol dipropionate | Agofollin | Estrogen | IM, SC | 2–10 mg/wk or 5–20 mg every 2 wks |
Estradiol benzoate | Progynon-B | Estrogen | IM, SC | 0.5–1.5 mg every 2–3 days |
Estriol | Ovestin [c] | Estrogen | Oral | 4–6 mg/day |
Spironolactone | Aldactone | Antiandrogen | Oral | 100–400 mg/day |
Cyproterone acetate | Androcur | Antiandrogen; Progestogen |
Oral | 5–100 mg/day |
Androcur Depot | IM | 300 mg/month | ||
Bicalutamide | Casodex | Antiandrogen | Oral | 25–50 mg/day |
Enzalutamide | Xtandi | Antiandrogen | Oral | 160 mg/day |
GnRH analogue | Various | GnRH modulator | Various | Variable |
Elagolix | Orilissa | GnRH antagonist | Oral | 150 mg/day or 200 mg twice daily |
Finasteride | Propecia | 5αR inhibitor | Oral | 1–5 mg/day |
Dutasteride | Avodart | 5αR inhibitor | Oral | 0.25–0.5 mg/day |
Progesterone | Prometrium [c] | Progestogen | Oral | 100–400 mg/day |
Medroxyprogesterone acetate | Provera | Progestogen | Oral | 2.5–40 mg/day |
Depo-Provera | Progestogen | IM | 150 mg every 3 mos | |
Depo-SubQ Provera 104 | Progestogen | SC | 104 mg every 3 mos | |
Hydroxyprogesterone caproate | Proluton | Progestogen | IM | 250 mg/wk |
Dydrogesterone | Duphaston | Progestogen | Oral | 20 mg/day |
Drospirenone | Slynd | Progestogen | Oral | 3 mg/day |
Domperidone [d] | Motilium | Prolactin releaser | Oral | 30–80 mg/day [e] |
|
When we prescribed estradiol, we preferred sublingual estradiol valerate instead of the oral form for feminizing HT since prior researchers have reported the effectiveness of sublingual administration in maintaining high blood estradiol concentration and low E1/E2 ratio [13].